September Publications

By Medicinal Chemistry Faculty, Students, and Researchers
Oct. 12, 2020

A Phosphoramidate Strategy Enables Membrane Permeability of a Non-nucleotide Inhibitor of the Prolyl Isomerase Pin1

Schwarz, D. M. C.;  Williams, S. K.;  Dillenburg, M.Wagner, C. R.; Gestwicki, J. E. ACS Med Chem Lett 2020, 11 (9), 1704-1710.

Comparative Intracerebroventricular and Intrathecal Administration of a Nanomolar Macrocyclic Melanocortin Receptor Agonist MDE6-5-2c (c[Pro-His-DPhe-Arg-Trp-Dap-Ala-DPro]) Decreases Food Intake in Mice
Adank, D. N.Lunzer, M. M.Ericson, M. D.Koeperich, Z. M.Wilber, S. L. Fleming, K. A.; Haskell-Luevano, C. ACS Chem Neurosci 2020, 11 (19), 3051-3063.

Development of small-molecule inhibitors of fatty acyl-AMP and fatty acyl-CoA ligases in Mycobacterium tuberculosis
Baran, M.;  Grimes, K. D.;  Sibbald, P. A.;  Fu, P.;  Boshoff, H. I. M.;  Wilson, D. J.; Aldrich, C. C., Eur J Med Chem 2020, 201, 112408.

DFG-1 Binding: A New Residue for Developing Selective Kinase Inhibitors
Faber, E. B.; Georg, G. I. J Med Chem 2020, 63 (18), 10221-10223.

Mass Spectrometric Quantitation of Apurinic/Apyrimidinic Sites in Tissue DNA of Rats Exposed to Tobacco-Specific Nitrosamines and in Lung and Leukocyte DNA of Cigarette Smokers and Nonsmokers
Guo, J.Chen, H.;  Upadhyaya, P.;  Zhao, Y.;  Turesky, R. J.; Hecht, S. S. Chem Res Toxicol 2020, 33 (9), 2475-2486.

ACS Medicinal Chemistry Letters Journal Cover, SeptemberACS Chemical Neuroscience Journal Cover, SeptemberEuropean Journal of Medicinal Chemistry Journal Cover, SeptemberACS Journal of Medicinal Chemistry Journal Cover, SeptemberChemical Research in Toxicology Journal Cover, September